Raloxifene 4'-glucuronide-d4 (lithium)
Catalog Number | Pack Size | List Price* | Quantity | |
---|---|---|---|---|
HY-135582S1-1MG | 1mg | Inquire | ||
HY-135582S1-5MG | 5mg | Inquire |
* CHF, excl. 8.1% VAT and shipping costs
Product Description
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Raloxifene 4'-glucuronide-d4 (lithium) is deuterium labeled Raloxifene 4'-glucuronide. Raloxifene 4'-glucuronide is a primary metabolite of Raloxifene. Raloxifene 4'-glucuronide formation is mediated mostly by UGT1A10 and UGT1A8. Raloxifene 4'-glucuronide binds to estrogen receptor with an IC50 of 370 μM. [1][2]. Raloxifene is a selective estrogen receptor modulator. Raloxifene activates TGFβ3 promoter as a full agonist at nanomolar concentrations, and inhibits the estrogen response element-containing vitellogenin promoter expression[3].
Category | Biochemicals |
Supplier | MedChem Express |
Application | Isotope-labeled compound |
Regulatory Status | RUO |
Research Field | Endocrinology, s,Vitamin D Related/Nuclear Receptor |
Format | Solubility: 10 mM in DMSO |
Grade | Clinical information: No Development Reported |
Molecular Formula | C34H30D4LiNO10S |
Molecular Weight | 659.67 |
Tech. Data Sheet | View datasheet |
Link To Supplier | http://www.medchemexpress.com |
Shipping Details | Room temperature |
Material Safety Data Sheet | Download PDF |