Relugolix-d6


Catalog Number Pack Size List Price* Quantity
HY-16474S-5MG 5mg   Inquire
HY-16474S-1MG 1mg   Inquire

* CHF, excl. 8.1% VAT and shipping costs


Product Description

Best price guarantee – we offer you the lowest price in Switzerland. Please contact us for a quote if needed.

Relugolix-d6 is deuterium labeled Relugolix. Relugolix (TAK-385) is a potent, orally active, nonpeptidic gonadotropin-releasing hormone (GnRH) antagonist. Relugolix possesses high affinity and potent antagonistic activity for human receptor (binding IC50=0.33 nM) and monkey receptor (IC50=0.32 nM) compared with TAK-013 (HY-100209)[1]. Relugolix is used for the study of sex-hormone-dependent diseases, such as including endometriosis, uterine fibroids and prostate cancer et al[2].

Category Biochemicals
Supplier MedChem Express
Application Isotope-labeled compound
Regulatory Status RUO
Research Field Cancer, Endocrinology, GPCR/G Protein,s
Format Solubility: 10 mM in DMSO
Grade Clinical information: No Development Reported
Molecular Formula C29H21D6F2N7O5S
Molecular Weight 629.67
Tech. Data Sheet View datasheet
Link To Supplier http://www.medchemexpress.com
Shipping Details Room temperature
Material Safety Data Sheet Download PDF