KDM5A-IN-1
| Catalog Number | Pack Size | List Price* | Quantity | |
|---|---|---|---|---|
| HY-100014-1MG | 1 mg | 204,00 | Add | |
| HY-100014-5MG | 5 mg | 456,00 | Add | |
| HY-100014-1ML | 10mM/1mL | 620,00 | Add | |
| HY-100014-10MG | 10 mg | 647,00 | Add | |
| HY-100014-50MG | 50 mg | 1'914,00 | Add | |
| HY-100014-100MG | 100 mg | 2'673,00 | Add |
* CHF, excl. 8.1% VAT and shipping costs
Product Description
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KDM5A-IN-1 is a potent, orally bioavailable pan-histone lysine demethylases 5 (KDM5) inhibitor with IC50s of 45 nM, 56 nM and 55 nM for KDM5A, KDM5B and KDM5C, respectively, and with an EC50 value of 960 nM for PC9 H3K4Me3. KDM5A-IN-1 is significantly less potent against other KDM5B enzymes (1A, 2B, 3B, 4C, 6A, 7B)[1].
| Category | Inhibitor |
| Supplier | MedChem Express |
| Regulatory Status | RUO |
| Research Field | Cancer, Epigenetics |
| Format | Solubility: DMSO : ≥ 50 mg/mL |
| Grade | Clinical information: No Development Reported |
| Purity | 99.95% |
| Molecular Formula | C15H22N4O2 |
| Molecular Weight | 290.36 |
| CAS-Number | 1905481-36-8 |
| Storage Conditions | -20°C, 3 years; 4°C, 2 years (Powder) |
| Tech. Data Sheet | View datasheet |
| Link To Supplier | http://www.medchemexpress.com |
| Shipping Details | Room Temperature |
| Material Safety Data Sheet | Download PDF |
