GSK484 (hydrochloride)

Catalog Number Pack Size List Price* Quantity
HY-100514-5MG 5 mg 254,00 Add
HY-100514-1ML 10mM/1mL 284,00 Add
HY-100514-10MG 10 mg 380,00 Add
HY-100514-25MG 25 mg 760,00 Add
HY-100514-S-1ST Sample   Inquire

* CHF, excl. 8.1% VAT and shipping costs

Product Description

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GSK484 hydrochloride is a selective and reversible peptidylarginine deiminase 4 (PAD4) inhibitor. GSK484 hydrochloride demonstrates high affinity binding to PAD4 with IC50s of 50 nM in the absence of Calcium. In the presence of 2 mM Calcium, notably lower potency (250 nM) is observed.

Category Biochemicals
Supplier MedChem Express
Regulatory Status RUO
Research Field Cancer, Inflammation/Immunology, Cardiovascular Disease, Epigenetics
Format Solubility: DMSO : 125 mg/mL (ultrasonic);H2O : 50 mg/mL (ultrasonic)
Grade Clinical information: No Development Reported
Purity 99.72%
Molecular Formula C27H32ClN5O3
Molecular Weight 510.03
CAS-Number 1652591-81-5
Storage Conditions 4°C (Powder, stored under nitrogen, away from moisture)
Tech. Data Sheet View datasheet
Link To Supplier
Shipping Details Room Temperature
Material Safety Data Sheet Download PDF