GSK484 (hydrochloride)
Catalog Number | Pack Size | List Price* | Quantity | |
---|---|---|---|---|
HY-100514-5MG | 5 mg | 254,00 | Add | |
HY-100514-1ML | 10mM/1mL | 284,00 | Add | |
HY-100514-10MG | 10 mg | 380,00 | Add | |
HY-100514-25MG | 25 mg | 760,00 | Add | |
HY-100514-S-1ST | Sample | Inquire |
* CHF, excl. 8.1% VAT and shipping costs
Product Description
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GSK484 hydrochloride is a selective and reversible peptidylarginine deiminase 4 (PAD4) inhibitor. GSK484 hydrochloride demonstrates high affinity binding to PAD4 with IC50s of 50 nM in the absence of Calcium. In the presence of 2 mM Calcium, notably lower potency (250 nM) is observed.
Category | Biochemicals |
Supplier | MedChem Express |
Regulatory Status | RUO |
Research Field | Cancer, Inflammation/Immunology, Cardiovascular Disease, Epigenetics |
Format | Solubility: DMSO : 125 mg/mL (ultrasonic);H2O : 50 mg/mL (ultrasonic) |
Grade | Clinical information: No Development Reported |
Purity | 99.72% |
Molecular Formula | C27H32ClN5O3 |
Molecular Weight | 510.03 |
CAS-Number | 1652591-81-5 |
Storage Conditions | 4°C (Powder, stored under nitrogen, away from moisture) |
Tech. Data Sheet | View datasheet |
Link To Supplier | http://www.medchemexpress.com |
Shipping Details | Room Temperature |
Material Safety Data Sheet | Download PDF |