Sigma-1 receptor antagonist 3


Catalog Number Pack Size List Price* Quantity
HY-125820-5MG 5 mg 393,00 Add
HY-125820-1ML 10mM/1mL 432,00 Add
HY-125820-10MG 10 mg 647,00 Add
HY-125820-50MG 50 mg 1'851,00 Add
HY-125820-100MG 100 mg 2'610,00 Add
HY-125820-S-1ST Sample   Inquire

* CHF, excl. 8.1% VAT and shipping costs


Product Description

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Sigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (σ1) receptor antagonist with a Ki of 1.14 nM. Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG) with an IC50 of 1.54 μM. Sigma-1 receptor antagonist 3 has the potential for the neuropathic pain[1].

Category Protein
Supplier MedChem Express
Regulatory Status RUO
Research Field Neurological Disease, Membrane Transporter/Ion Channel,Neuronal Signaling
Format Solubility: DMSO : 12.5 mg/mL (ultrasonic)
Grade Clinical information: No Development Reported
Purity 99.47%
Molecular Formula C19H23ClFN3O
Molecular Weight 363.86
CAS-Number 1639220-17-9
Storage Conditions -20°C, 3 years; 4°C, 2 years (Powder)
Tech. Data Sheet View datasheet
Link To Supplier http://www.medchemexpress.com
Shipping Details Room Temperature
Material Safety Data Sheet Download PDF