BMS-986202
| Catalog Number | Pack Size | List Price* | Quantity | |
|---|---|---|---|---|
| HY-131968-5MG | 5mg | 521,00 | Add | |
| HY-131968-1ML | 10mM/1mL | 571,00 | Add | |
| HY-131968-10MG | 10 mg | 925,00 | Add | |
| HY-131968-25MG | 25 mg | 1'786,00 | Add | |
| HY-131968-50MG | 50 mg | 2'801,00 | Add | |
| HY-131968-100MG | 100 mg | 4'320,00 | Add |
* CHF, excl. 8.1% VAT and shipping costs
Product Description
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BMS-986202 is a potent, selective and orally active Tyk2 inhibitor that binds to Tyk2 JH2 with an IC50 value of 0.19 nM and a Ki of 0.02 nM. BMS-986202 is remarkably selective over other kinases including Jak family members. BMS-986202 is also a weak inhibitor of CYP2C19 with an IC50 value of 14 μM. BMS-986202 can be used for IL-23-driven acanthosis, anti-CD40-induced colitis, and spontaneous lupus research. BMS-986202 is a de novo deuterium[1].
| Category | Biochemicals |
| Supplier | MedChem Express |
| Application | Isotope-labeled compound |
| Regulatory Status | RUO |
| Research Field | Inflammation/Immunology, Epigenetics,JAK/STAT Signaling,Metabolic Enzyme/Protease,Protein Tyrosine Kinase/RTK,Stem Cell/Wnt |
| Format | Solubility: DMSO : 250 mg/mL (ultrasonic) |
| Grade | Clinical information: Phase 1 |
| Purity | 99.92% |
| Molecular Formula | C22H18D3FN6O3 |
| Molecular Weight | 439.46 |
| CAS-Number | 1771691-34-9 |
| Storage Conditions | -20°C, 3 years; 4°C, 2 years (Powder) |
| Tech. Data Sheet | View datasheet |
| Link To Supplier | http://www.medchemexpress.com |
| Shipping Details | Room Temperature |
| Material Safety Data Sheet | Download PDF |
