Enpatoran
| Catalog Number | Pack Size | List Price* | Quantity | |
|---|---|---|---|---|
| HY-134581-1MG | 1 mg | 204,00 | Add | |
| HY-134581-5MG | 5 mg | 393,00 | Add | |
| HY-134581-10MG | 10 mg | 584,00 | Add | |
| HY-134581-25MG | 25 mg | 989,00 | Add | |
| HY-134581-50MG | 50 mg | 1'470,00 | Add | |
| HY-134581-100MG | 100 mg | 2'142,00 | Add | |
| HY-134581-200MG | 200 mg | 3'118,00 | Add |
* CHF, excl. 8.1% VAT and shipping costs
Product Description
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Enpatoran (M5049) is a potent, orally active and dual TLR7/8 inhibitor with IC50s of 11.1 nM and 24.1 nM in HEK293 cells, respectively. Enpatoran is inactive against TLR3, TLR4 and TLR9. Enpatoran can block molecule synthetic ligands and natural endogenous RNA ligands. Enpatoran exhibits excellent pharmacokinetic properties in vivo. Enpatoran can be used for both innate and adaptive autoimmunity blocking research [1].
| Category | Biochemicals |
| Supplier | MedChem Express |
| Regulatory Status | RUO |
| Research Field | Inflammation/Immunology, Immunology/Inflammation |
| Format | Solubility: DMSO : 24.44 mg/mL (ultrasonic);Ethanol : 100 mg/mL (ultrasonic) |
| Grade | Clinical information: Phase 2 |
| Purity | 99.77% |
| Molecular Formula | C16H15F3N4 |
| Molecular Weight | 320.31 |
| CAS-Number | 2101938-42-3 |
| Storage Conditions | -20°C (Powder, sealed storage, away from moisture and light) |
| Tech. Data Sheet | View datasheet |
| Link To Supplier | http://www.medchemexpress.com |
| Shipping Details | Blue Ice |
| Material Safety Data Sheet | Download PDF |
