KDM5A-IN-1 (Standard)
| Catalog Number | Pack Size | List Price* | Promo Price* | Quantity | |
|---|---|---|---|---|---|
| HY-100014R-1MG | 1 mg | 382,00 | 236,90 | Add | |
| HY-100014R-5MG | 5 mg | 924,00 | 572,90 | Add | |
| HY-100014R-10MG | 10 mg | 1'377,00 | 853,80 | Add | |
| HY-100014R-25MG | 25 mg | 2'462,00 | 1'526,50 | Add | |
| HY-100014R-50MG | 50 mg | 3'682,00 | 2'282,90 | Add | |
| HY-100014R-100MG | 100 mg | 5'509,00 | 3'415,60 | Add |
* CHF, excl. 8.1% VAT and shipping costs
Product Description
Promotion runs until 31.12.2026Best price guarantee – we offer you the lowest price in Switzerland. Please contact us for a quote if needed.
KDM5A-IN-1 (Standard) is the analytical standard of KDM5A-IN-1 (HY-100014) . This product is intended for research and analytical applications. KDM5A-IN-1 is a potent, orally bioavailable pan-histone lysine demethylases 5 (KDM5) inhibitor with IC50s of 45 nM, 56 nM and 55 nM for KDM5A, KDM5B and KDM5C, respectively, and with an EC50 value of 960 nM for PC9 H3K4Me3. KDM5A-IN-1 is significantly less potent against other KDM5B enzymes (1A, 2B, 3B, 4C, 6A, 7B) [1].
| Category | Inhibitor |
| Supplier | MedChem Express |
| Regulatory Status | RUO |
| Research Field | Cancer |
| Molecular Formula | C15H22N4O2 |
| Molecular Weight | 290.37 |
| CAS-Number | 1905481-36-8 |
| Tech. Data Sheet | View datasheet |
| Link To Supplier | http://www.medchemexpress.com |
| Shipping Details | Room temperature |
| Material Safety Data Sheet | Download PDF |
